Cabergoline
D2-like receptor agonistProduct Code: Asc-564 |
Purity: >99% |
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| Buy Cabergoline from Abcam | ||||
Biological DescriptionD2-like receptor agonist (Ki values are 0.7, 1.5, 9.0 and 165 nM at D2, D3, D4 and D5 receptors respectively). Highly potent at some 5-HT receptors (Ki values are 20, 8.7, 6.2 and 1.2 nM at 5-HT1A, 5-HT1D, 5-HT2A and 5-HT2B respectively). Shows anti-tumour effects and has anti-depressant and anxiolytic properties. |
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Useful References | |
Cabergoline, a dopamine receptor agonist, has an antidepressant-like property and enhances brain-derived neurotrophic factor signaling. abstract A review of the receptor-binding and pharmacokinetic properties of dopamine agonists. abstract In vivo effect of cabergoline, a dopamine agonist, on estrogen-induced rat pituitary tumors. abstract | |
Chemical InformationN-[3-(Dimethylamino)propyl]-N-[(ethylamino)carbonyl]-6-(2-propenyl)ergoline-8β-carboxamide | |
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