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Endomorphin-1

Highly potent and selective μ agonist

Product Code: Asc-411

Purity: >98%

  
Pack Size

 

5mg
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Biological Description

Endogenous peptide with extremely high affinity for μ opioid receptors (Ki = 360 pM). Displays 4000- and 15000-fold selectivity over δ and κ receptors respectively.
Useful References

(1997) A potent and selective endogenous agonist for the µ-opiate receptor. Nature 386:499-502 abstract

(1998) Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J.Pharmacol Exp Ther 286;1007-13. abstract

(2000) Endomorphin-1 and endomorphin-2: pharmacology of the selective endogenous mu-opioid receptor agonists. Pharmacol Ther. 88:437-63. abstract

Chemical Information

YPWF-NH2

Asc-411
  • Desiccate at -20°C
  • MW 610.67
  • Soluble in water
  • C34H38N6O5
  • 189388-22-5