Home > Enzymes > Kinase
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Product Purity Feature Pack
8-Br-cAMP (8-Bromo-cAMP)
Code: Asc-1448
cAMP analog. PKA activator.
>98%  
5mg
25mg
Buy from Abcam
A 83-01
Code: Asc-2092
Potent ALK4, 5 and 7 kinase inhibitor
>98%  
1mg
5mg
Buy from Abcam
A 769662
Code: Asc-335
AMP-activated protein kinase activator
>99%  
10mg
50mg
Buy from Abcam
AAL-993
Code: Asc-1590
Potent, selective and cell-permeable VEGFR inhibitor
>98%  
5mg
25mg
Buy from Abcam
Adenosine 3′,5′-cyclic monophosphate (cAMP)
Code: Asc-493
Second messenger. PKA activator.
>98%  
1g
5g
25g
Buy from Abcam
AG-370
Code: Asc-1563
Selective PDGFR tyrosine kinase inhibitor
>99%  
2mg
10mg
Buy from Abcam
AG-494
Code: Asc-1562
Potent, selective EGF receptor tyrosine kinase
>99%  
10mg
Buy from Abcam
AG 1296
Code: Asc-1170
Potent specific PDGF receptor tyrosine kinase inhibitor
>99%  
5mg
25mg
Buy from Abcam
AG 1478
Code: Asc-1438
Selective EGF receptor tyrosine kinase inhibitor
>98%  
5mg
25mg
Buy from Abcam
AG 490
Code: Asc-950
JAK2/3 inhibitor
>99%  
10mg
50mg
Buy from Abcam
AG-879
Code: Asc-1059
Selective TrkA receptor inhibitor
>99%  
10mg
Buy from Abcam
AICAR (Acadesine/AICA riboside)
Code: Asc-358
Cell-permeable activator of AMP-activated protein kinase
>98%  
50mg
250mg
Buy from Abcam
Akt Inhibitor, Isozyme-Selective
Code: Asc-2088
Potent isozyme selective Akt1/2 kinase inhibitor
>97%  
1mg
Buy from Abcam
Alsterpaullone
Code: Asc-1070
Potent cyclin-dependent kinase (CDK) and GSK-3β inhibitor
>99%  
1mg
Buy from Abcam
Anisomycin
Code: Asc-495
Protein synthesis inhibitor
>98%  
10mg
50mg
Buy from Abcam
AR-A014418
Code: Asc-1295
Highly selective GSK-3 inhibitor
>99%  
10mg
50mg
Buy from Abcam
AS-041164
Code: Asc-898
Potent and selective PI3Kγ inhibitor
>98%  
5mg
25mg
Buy from Abcam
AS-252424
Code: Asc-929
Potent and selective PI3Kγ inhibitor
>95%  
5mg
10mg
Buy from Abcam
AS-604850
Code: Asc-935
Selective, ATP-competitive PI3Kγ inhibitor
>98%  
5mg
25mg
Buy from Abcam
AS-605240
Code: Asc-928
Potent and selective PI3Kγ inhibitor
>98%  
10mg
50mg
Buy from Abcam
AT9283
Code: Asc-1341
Potent Aurora A and B kinase inhibitor
>95%  
10mg
50mg
Buy from Abcam
AZ-960
Code: Asc-1342
Novel, potent and selective JAK2 inhibitor
>95%  
1mg
5mg
Buy from Abcam
AZD1152-HQPA
Code: Asc-2049
Potent, selective Aurora B kinase inhibitor
>99%  
5mg
25mg
Buy from Abcam
AZD7762
Code: Asc-1344
Novel checkpoint kinase inhibitor
>95%  
10mg
50mg
Buy from Abcam
Bay 61-3606 hydrochloride
Code: Asc-2106
Potent, selective, cell-permeable Syk kinase inhibitor
>98%  
1mg
5mg
Buy from Abcam
BIBW2992 (Afatinib)
Code: Asc-2064
Potent, irreversible ATP-competitive ErbB inhibitor. Antitumor.
>99%  
1mg
5mg
Buy from Abcam
Bikinin
Code: Asc-2203
Cell-permeable, ATP-competitive 7 Arabidopsis GSK-3 inhibitor
>95%  
10mg
50mg
Buy from Abcam
BIO
Code: Asc-891
Potent, selective, reversible GSK3 inhibitor; cell-permeable
>98%  
10mg
25mg
Buy from Abcam
BML-259
Code: Asc-1585
Potent Cdk5/p25 and Cdk2 inhibitor
>98%  
5mg
25mg
Buy from Abcam
BMS-599626 (AC480)
Code: Asc-2063
Selective HER1 and HER2 inhibitor
>99%  
1mg
5mg
Buy from Abcam
Bosutinib (SKI-606)
Code: Asc-1987
Potent dual Abl and selective Src kinase inhibitor
   
10mg
50mg
Buy from Abcam
Butyrolactone I
Code: Asc-1520
Cell permeable, selective, ATP-competitive cyclin-dependent kinase (CDK) inhibitor
>99%  
200µg
1mg
Buy from Abcam
Canertinib (CI-1033)
Code: Asc-1402
Potent irreversible EGFR and HER2/ErbB2 tyrosine kinase inhibitor
>99%  
5mg
50mg
Buy from Abcam
CAY10505
Code: Asc-930
Potent PI3Kγ and casein kinase 2 inhibitor
>98%  
10mg
50mg
Buy from Abcam
CAY10577
Code: Asc-944
CK2 inhibitor
>95%  
10mg
50mg
Buy from Abcam
CAY10578
Code: Asc-945
Selective, ATP competitive CK2 inhibitor
>95%  
5mg
25mg
Buy from Abcam
CAY10626
Code: Asc-903
Potent PI3Kα/mTOR inhibitor
>98%  
1mg
5mg
Buy from Abcam
Celastrol from Celastrus scandens
Code: Asc-655
Anti-inflammatory and anti-proliferative agent
>99%  
10mg
50mg
Buy from Abcam
CGP 57380
Code: Asc-365
MNK inhibitor
>98%  
1mg
10mg
50mg
Buy from Abcam
Chelerythrine chloride
Code: Asc-600
Apoptosis inducer. Protein kinase C inhibitor.
>99%  
5mg
Buy from Abcam
CHIR99021
Code: Asc-890
Potent, highly selective GSK3 inhibitor
>98%  
1mg
5mg
Buy from Abcam
Chk2 inhibitor
Code: Asc-2086
Potent, ATP-competitive checkpoint kinase (Chhk) 2 inhibitor. Cell-permeable.
>98%  
1mg
Buy from Abcam
8-(4-Chlorophenylthio)adenosine 3',5'-cyclic monophosphate (8-CPT-cAMP)
Code: Asc-424
Cell permeable cAMP analogue, protein kinase modulator
>98%  
20mg
100mg
Buy from Abcam
CI-1040
Code: Asc-1348
ATP non-competitive MEK1/2 inhibitor
>95%  
10mg
50mg
Buy from Abcam
Compound 401
Code: Asc-968
Selective, reversible DNA-dependent protein kinase and mTOR inhibitor
>99%  
10mg
50mg
Buy from Abcam
CP-724714
Code: Asc-1349
Potent, selective HER2/ErbB2 tyrosine kinase inhibitor
>95%  
10mg
50mg
Buy from Abcam
Crosstide
Code: Asc-964
Akt peptide substrate
>98%  
1mg
Buy from Abcam
Crosstide (biotinylated)
Code: Asc-965
Akt peptide substrate, biotinylated
>98%  
1mg
Buy from Abcam
CX-4945 (Silmitasertib)
Code: Asc-1350
Potent, selective ATP-competitive casein kinase 2 inhibitor
>95%  
1mg
5mg
Buy from Abcam
D4476
Code: Asc-220
CK1 inhibitor
>99%  
10mg
50mg
Buy from Abcam
Dasatinib
Code: Asc-2050
Protein kinase inhibitor. Anti-tumor.
>99%  
25mg
100mg
Buy from Abcam
(-)-Deguelin
Code: Asc-941
Akt inhibitor. Anti-cancer agent.
>98%  
10mg
50mg
Buy from Abcam
DL-threo-Dihydrosphingosine
Code: Asc-1753
Potent sphingosine kinase inhibitor
>98%  
10mg
50mg
Buy from Abcam
7,8-Dihydroxyflavone (7,8-DHF)
Code: Asc-996
Selective TrkB receptor agonist. Flavonoid.
>99%  
10mg
50mg
Buy from Abcam
DMPQ dihydrochloride
Code: Asc-1269
Potent and selective PDGFRβ inhibitor
>99%  
10mg
50mg
Buy from Abcam
Dorsomorphin
Code: Asc-843
Potent, selective and reversible AMP-kinase inhibitor. Selective for BMP signaling.
>99%  
10mg
50mg
Buy from Abcam
DRB (Benzimidazole)
Code: Asc-939
Casein kinase II inhibitor
>98%  
10mg
50mg
Buy from Abcam
E6 Berbamine
Code: Asc-1519
Selective, cell-permeable calmodulin (CaM) antagonist
>98%  
10mg
50mg
Buy from Abcam
Ellagic acid
Code: Asc-622
Selective, casein kinase 2 (CK2) inhibitor
>99%  
50mg
Buy from Abcam
(-)-Epigallocatechin Gallate
Code: Asc-716
Potent anti-oxidant flavonoid
>98%  
1mg
50mg
Buy from Abcam
Erbstatin Analog
Code: Asc-1549
EGFR tyrosine kinase inhibitor
>98%  
5mg
25mg
Buy from Abcam
Erlotinib (CP-358,774)
Code: Asc-881
Potent, selective and reversible EGFR tyrosine kinase inhibitor
>98%  
250mg
1g
Buy from Abcam
Erlotinib hydrochloride
Code: Asc-1930
Potent HER-1/EGFR tyrosine kinase inhibitor
>98%  
10mg
25mg
100mg
500mg
Buy from Abcam
Everolimus
Code: Asc-2151
Potent mTOR inhibitor
>98%  
5mg
25mg
Buy from Abcam
Farnesyl thiotriazole
Code: Asc-1706
Stable, potent PKC activator
>98%  
10mg
50mg
Buy from Abcam
Gambogic amide
Code: Asc-1702
Potent, selective high affinity nerve growth factor (TrKa) receptor agonist
>98%  
1mg
5mg
Buy from Abcam
GDC-0941
Code: Asc-1352
Potent, non-selective PI3K inhibitor
>95%  
10mg
50mg
Buy from Abcam
Genistein
Code: Asc-112
Protein tyrosine kinase inhibitor. Anticancer agent.
>99%  
10mg
50mg
100mg
Buy from Abcam
Genistin
Code: Asc-1395
Isoflavone glycoside; inactive analog of Genistein
>99%  
10mg
Buy from Abcam
GF 109203X HCl
Code: Asc-844
Potent, cell permeable, ATP-competitive PKC inhibitor
>99%  
1mg
10mg
Buy from Abcam
[Ala19]-Glucagon-Like Peptide II (rat)
Code: Asc-2239
Intestinal growth factor
   
0
500µg
1mg
2.5mg
Buy from Abcam
Go 6976
Code: Asc-1413
Potent PKC inhibitor. Selective for PKCα and β
>99%  
500µg
Buy from Abcam
GW2580
Code: Asc-2096
Selective cFMS RTK inhibitor. Cell-permeable.
>99%  
5mg
25mg
Buy from Abcam
H89 dihydrochloride
Code: Asc-341
Kinase inhibitor
>98%  
1mg
10mg
50mg
Buy from Abcam
HA-1077 (Fasudil)
Code: Asc-306
ROCK2 inhibitor
>98%  
10mg
50mg
Buy from Abcam
Harmine
Code: Asc-225
Potent and selective inhibitor of DYRK1A
>98%  
100mg
Buy from Abcam
HBDDE
Code: Asc-1573
Selective PKCα and PKCγ inhibitor
>97%  
1mg
5mg
Buy from Abcam
1-O-Hexadecyl-2-O-acetyl-sn-glycerol
Code: Asc-1550
Protein Kinase C Inhibitor. DAG analog
>95%  
5mg
Buy from Abcam
Hydralazine hydrochloride
Code: Asc-863
DNA methylation inhibitor. Anti-hypertensive agent
>99%  
1g
Buy from Abcam
HNMPA-(AM)3
Code: Asc-1567
Insulin receptor tyrosine kinase inhibitor
>98%  
5mg
25mg
Buy from Abcam
IKK-ε Kinase Inhibitor II
Code: Asc-2109
Inhibitor of IκB kinases (IKK)
>97%  
1mg
5mg
Buy from Abcam
Indirubin
Code: Asc-960
Potent cyclin-dependent kinase and GSK-3β inhibitor
>98%  
5mg
25mg
Buy from Abcam
Iodotubercidin
Code: Asc-452
Potent, adenosine kinase inhibitor
>95%  
1mg
5mg
Buy from Abcam
IPA 3
Code: Asc-1014
Group I, p21-activated kinase (PAK) inhibitor
>97%  
10mg
50mg
Buy from Abcam
Isobavachalcone
Code: Asc-1168
Akt inhibitor. Natural chalcone.
>99%  
1mg
Buy from Abcam
Isoprenaline hydrochloride
Code: Asc-710
Non selective β-adrenoceptor agonist
>99%  
100mg
Buy from Abcam
K252a
Code: Asc-419
Highly potent inhibitor of protein and CAM kinases
>99%  
200µg
1mg
Buy from Abcam
Kenpaullone
Code: Asc-937
CDK2, GSK3β and LCK inhibitor
>98%  
5mg
10mg
Buy from Abcam
Ki20227
Code: Asc-1357
Highly selective c-Fms tyrosine kinase inhibitor
>95%  
10mg
50mg
Buy from Abcam
KN-62
Code: Asc-421
CaM kinase II inhibitor. P2X7 antagonist.
>98%  
1mg
5mg
Buy from Abcam
KN-93 (water soluble)
Code: Asc-980
Potent, specific CaMK II inhibitor
>99%  
1mg
Buy from Abcam
KT5823
Code: Asc-423
Potent, selective inhibitor of PKG
>95%  
100µg
Buy from Abcam
KU-55933
Code: Asc-637
Potent, selective, competitive ATM kinase inhibitor
>99%  
10mg
Buy from Abcam
L803
Code: Asc-966
Phosphopeptide GSK-3 inhibitor
>99%  
1mg
Buy from Abcam
Lapatinib Ditosylate (Tykerb)
Code: Asc-2069
Potent ErbB-2 and EGFR dual tyrosine kinase inhibitor. Antitumor.
>99%  
25mg
100mg
Buy from Abcam
Lavendustin A
Code: Asc-1556
Potent, selective tyrosine kinase inhibitor
>98%  
1mg
Buy from Abcam
Lavendustin B
Code: Asc-1570
Tyrosine kinase inhibitor
>98%  
5mg
Buy from Abcam
Lavendustin C
Code: Asc-1564
Potent EGF receptor tyrosine kinase inhibitor
>98%  
10mg
Buy from Abcam
LDN193189
Code: Asc-2186
Potent, selective ALK2 and ALK3 inhibitor
>97%  
5mg
25mg
Buy from Abcam
Lestaurtinib
Code: Asc-2107
Potent JAK2, FLT3 and TrkA receptor tyrosine kinase inhibitor
>98%  
500µg
1mg
Buy from Abcam
LFM-A13
Code: Asc-1575
Selective BTK inhibitor
>97%  
5mg
Buy from Abcam
Lithium chloride
Code: Asc-853
GSK-3β inhibitor
>99%  
1g
5g
Buy from Abcam
Luteolin
Code: Asc-662
Antioxidant, anti-inflammatory, anti-cancer flavonoid
>99%  
10mg
50mg
Buy from Abcam
LY 294002
Code: Asc-243
PI3-kinase inhibitor
>99%  
5mg
25mg
Buy from Abcam
LY 303511 dihydrochloride
Code: Asc-956
Negative control for LY 294002 (Asc-243)
>98%  
5mg
Buy from Abcam
Metformin hydrochloride
Code: Asc-847
AMPK activator
>99%  
100mg
Buy from Abcam
2-Methoxyestradiol
Code: Asc-653
Potent antitumor and antiangiogenic agent
>98%  
10mg
50mg
Buy from Abcam
ML7
Code: Asc-848
Potent, selective myosin light chain kinase inhibitor
>99%  
10mg
50mg
Buy from Abcam
Momelotinib
Code: Asc-1372
Selective JAK2 inhibitor
>95%  
10mg
50mg
Buy from Abcam
MS-1020
Code: Asc-1465
Selective, cell-permeable JAK3 inhibitor
>95%  
1mg
Buy from Abcam
Myricetin
Code: Asc-721
Potent anti-neoplastic, anti-oxidant and anti-inflammatory agent
>97%  
5mg
25mg
Buy from Abcam
Hydroxy-2-naphthalenylmethylphosphonic acid (HNMPA)
Code: Asc-1566
Insulin receptor tyrosine kinase inhibitor
>98%  
5mg
25mg
Buy from Abcam
Nifuroxazide
Code: Asc-951
JAK/STAT signaling inhibitor. Nitrofuran antibiotic.
>98%  
100mg
Buy from Abcam
Nimbolide
Code: Asc-2138
CyclinA and ERK1/2 inhibitor. Terpenoid lactone.
>98%  
5mg
25mg
Buy from Abcam
NSC 210902
Code: Asc-943
Selective, ATP competitive CK2 inhibitor
>95%  
10mg
50mg
Buy from Abcam
NU 7026
Code: Asc-970
Novel, specific, reversible DNA-PK inhibitor
>99%  
10mg
50mg
Buy from Abcam
NVP-BSK805
Code: Asc-1373
Selective JAK2 inhibitor
>95%  
10mg
50mg
Buy from Abcam
Olomoucine
Code: Asc-938
ATP-competitive CDK inhibitor
>98%  
5mg
25mg
Buy from Abcam
Olomoucine II
Code: Asc-1238
CDK/cyclin inhibitor
>98%  
1mg
5mg
Buy from Abcam
P1
Code: Asc-2325
Inhibits EGF receptor binding to SH2 of phospholipase Cγ1.
   
0
500µg
1mg
2.5mg
Buy from Abcam
1-O-Palmitoyl-2-O-acetyl-sn-glycero-3-phosphorylcholine
Code: Asc-1684
Platelet activating factor (PAF) agonist
>99%  
1mg
5mg
Buy from Abcam
Palmitoyl-L-carnitine chloride
Code: Asc-2334
Protein kinase inhibitor
>98%  
5mg
10mg
Buy from Abcam
(±)-Palmitoylcarnitine chloride
Code: Asc-1122
Protein kinase C (PKC) inhibitor. Intermediate in lipid metabolism.
>98%  
100mg
Buy from Abcam
PD 153035 Hydrochloride
Code: Asc-2076
Highly potent, selective EGFR tyrosine kinase inhibitor
>95%  
2mg
Buy from Abcam
PD 0325901
Code: Asc-639
Potent MEK 1 and 2 inhibitor
>99%  
10mg
50mg
Buy from Abcam
PD 173074
Code: Asc-1117
Potent FGFR1 and FGFR3 inhibitor
>99%  
10mg
50mg
Buy from Abcam
PD 98059
Code: Asc-234
MEK1 inhibitor
>99%  
1mg
10mg
50mg
Buy from Abcam
Pelitinib (EKB-569)
Code: Asc-1171
Irreversible EGFR inhibitor
>98%  
5mg
25mg
Buy from Abcam
Perifosine
Code: Asc-2055
Akt inhibitor; alkylphospholipid
>99%  
5mg
25mg
Buy from Abcam
Perillyl alcohol
Code: Asc-2452
Natural monoterpene
>85%  
10g
50g
Buy from Abcam
PF-04691502
Code: Asc-2009
Potent, selective ATP-competitive dual PI3K/mTOR inhibitor
   
10mg
50mg
Buy from Abcam
PF-4708671
Code: Asc-1993
Potent, selective, cell-permeable p70 ribosomal S6 kinase inhibitor
   
10mg
50mg
Buy from Abcam
PF431396
Code: Asc-1359
Potent dual FAK/Pyk2 inhibitor
>95%  
1mg
5mg
Buy from Abcam
PF-562271
Code: Asc-1360
Potent, reversible, ATP-competitive FAK/Pyk2 inhibitor
>95%  
1mg
5mg
Buy from Abcam
PF 670462
Code: Asc-985
Potent, selective casein kinase 1ε (CK1ε) and CK1δ inhibitor
>99%  
10mg
50mg
Buy from Abcam
Phenformin hydrochloride
Code: Asc-1459
AMPK activator
>97%  
100mg
1g
Buy from Abcam
Phorbol 12-myristate 13-acetate (PMA)
Code: Asc-297
PKC activator
>99%  
1mg
5mg
25mg
Buy from Abcam
Phosphate Acceptor Peptide (Arg-Arg-Lys-Ala-Ser-Gly-Pro-Pro-Val)
Code: Asc-2346
PKC and S6 kinase substrate
   
1mg
2mg
5mg
Buy from Abcam
Phospho-Glycogen Synthase Peptide-2
Code: Asc-079
GSK substrate
>99%  
500µg
1mg
Buy from Abcam
PI 103
Code: Asc-1361
Novel, potent, ATP-competitive PI3K, mTOR and DNA-PK inhibitor
>95%  
10mg
50mg
Buy from Abcam
Piceatannol
Code: Asc-722
Syk tyrosine kinase inhibitor
>99%  
10mg
50mg
Buy from Abcam
PIK-75
Code: Asc-931
Selective p110α PI3K inhibitor
>98%  
5mg
25mg
Buy from Abcam
PKC412
Code: Asc-1494
Broad spectrum protein kinase inhibitor
>98%  
1mg
5mg
Buy from Abcam
PLX4720
Code: Asc-1362
Potent, selective mutant B-RafV600E and c-Raf-1Y340D/Y341D inhibitor
>95%  
10mg
50mg
Buy from Abcam
PP 1
Code: Asc-859
Potent Src family tyrosine kinase inhibitor
>98%  
10mg
Buy from Abcam
PP2
Code: Asc-308
Src and RIP2 kinase inhibitor
>98%  
1mg
5mg
10mg
Buy from Abcam
PP242
Code: Asc-1405
Potent and selective mTOR inhibitor
>98%  
1mg
Buy from Abcam
PP3
Code: Asc-617
Negative control for the Src kinase inhibitor PP2.
>98%  
10mg
100mg
Buy from Abcam
Prostratin
Code: Asc-880
PKC activator; reactivates HIV-1 latency
>98%  
500µg
1mg
Buy from Abcam
PS48
Code: Asc-2133
Allosteric phosphoinositide-dependent protein kinase-1 (PDK1) agonist
>95%  
5mg
25mg
Buy from Abcam
Purvalanol A
Code: Asc-304
Potent CDK inhibitor
>98%  
1mg
10mg
50mg
Buy from Abcam
Purvalanol B
Code: Asc-305
CDK2 inhibitor
>98%  
10mg
50mg
Buy from Abcam
Quizartinib
Code: Asc-2189
Potent, selective Flt3 inhibitor
>99%  
1mg
5mg
Buy from Abcam
RG-14620
Code: Asc-1569
EGF receptor tyrosine kinase inhibitor
>99%  
5mg
Buy from Abcam
Ro 31-8220 mesylate (Bisindolylmaleimide IX)
Code: Asc-374
Protein kinase inhibitor
>98%  
1mg
10mg
50mg
Buy from Abcam
RO-3306
Code: Asc-1491
Selective cyclin-dependent kinase (Cdk1) inhibitor
>95%  
1mg
5mg
Buy from Abcam
Rottlerin
Code: Asc-377
Kinase inhibitor
>90%  
10mg
50mg
Buy from Abcam
RR-SRC
Code: Asc-2363
Synthetic tyrosine kinase substrate
   
5mg
10mg
25mg
Buy from Abcam
SAMS peptide
Code: Asc-182
AMP-activated protein kinase substrate
>95%  
1mg
5mg
Buy from Abcam
SB 202190
Code: Asc-638
Highly selective, potent, cell permeable p38 MAP kinase inhibitor
>99%  
10mg
50mg
Buy from Abcam
SB 203580
Code: Asc-162
p38 MAP kinase inhibitor
>99%  
1mg
10mg
50mg
Buy from Abcam
SB 203580 hydrochloride
Code: Asc-235
p38 MAP kinase inhibitor; water soluble
>99%  
10mg
Buy from Abcam
SB 216763
Code: Asc-202
Potent selective GSK-3 inhibitor
>98%  
1mg
10mg
50mg
Buy from Abcam
SB 415286
Code: Asc-962
Potent, selective GSK-3 inhibitor
>99%  
10mg
50mg
Buy from Abcam
SB431542
Code: Asc-163
ALK inhibitor
>99%  
1mg
5mg
10mg
Buy from Abcam
SC-66
Code: Asc-802
Allosteric Akt inhibitor
>99%  
10mg
50mg
Buy from Abcam
SD 169
Code: Asc-836
Potent, selective and ATP competitive p38α MAPK inhibitor
>99%  
10mg
50mg
Buy from Abcam
SH-5
Code: Asc-1442
Specific Akt inhibitor
>98%  
500µg
Buy from Abcam
SH-6
Code: Asc-1443
Phosphatidylinositol analog; selective Akt inhibitor
>98%  
500µg
Buy from Abcam
SKI-I, Sphingosine Kinase Inhibitor
Code: Asc-2209
Specific non-lipid sphingosine kinase (SK) inhibitor. Cell-permeable.
>90%  
5mg
25mg
Buy from Abcam
SKI-II
Code: Asc-1594
Sphingosine kinase (SK1/2) inhibitor
>98%  
10mg
Buy from Abcam
SL 327
Code: Asc-082
MEK inhibitor
>99%  
1mg
10mg
25mg
Buy from Abcam
Sodium salicylate
Code: Asc-746
Cell permeable anti-inflammatory agent
>99%  
5g
Buy from Abcam
SP600125
Code: Asc-065
JNK inhibitor
>98%  
10mg
50mg
Buy from Abcam
Src Kinase Inhibitor I (SKI-1)
Code: Asc-839
Potent, selective and dual site Src tyrosine kinase family inhibitor
>98%  
10mg
50mg
Buy from Abcam
Staurosporine
Code: Asc-056
Protein kinase inhibitor
>98%  
100µg
500µg
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1-Stearoyl-2-arachidonoyl-sn-glycerol
Code: Asc-1530
Endogenous PKC activator
>98%  
10mg
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STO-609
Code: Asc-1591
Potent, competitive, selective and cell-permeable inhibitor of CaM-KK
>98%  
5mg
25mg
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SU 11274
Code: Asc-2159
Potent, selective cell-permeable Met inhibitor
>98%  
5mg
25mg
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SU 6668
Code: Asc-2156
Potent PDGFR inhibitor
>98%  
5mg
25mg
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SU 1498
Code: Asc-1447
Selective VEGFR2 inhibitor
>98%  
1mg
5mg
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SU4312
Code: Asc-1577
Potent, selective VEGFR and PDGFR receptor tyrosine kinase inhibitor
>98%  
5mg
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SU-5402
Code: Asc-1368
Potent FGFR and VEGFR inhibitor
>95%  
1mg
5mg
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Sulindac sulfide
Code: Asc-650
Active metabolite of Sulindac. COX-1/ 2 inhibitor.
>98%  
5mg
25mg
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TAK 165
Code: Asc-1473
Potent HER2 tyrosine kinase inhibitor
>98%  
5mg
25mg
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TAK 715
Code: Asc-989
Potent p38 MAPK inhibitor
>99%  
10mg
50mg
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TBB
Code: Asc-988
Selective, cell-permeable casein kinase-2 (CK2) inhibitor
>98%  
10mg
50mg
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TCS 359
Code: Asc-1268
Potent FLT3 receptor tyrosine kinase inhibitor
>99%  
10mg
50mg
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TCS JNK 5a
Code: Asc-835
Selective JNK2/3 inhibitor
>99%  
10mg
50mg
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TDZD-8
Code: Asc-2372
Selective, non-ATP competitive GSK-3β inhibitor
>98%  
5mg
25mg
100mg
250mg
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Temsirolimus
Code: Asc-1999
Selective mTOR inhibitor (IC50 = 1.76 µM).
   
10mg
50mg
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TG003
Code: Asc-1463
Potent, specific Cdc2-like (Clk) kinase inhibitor
>98%  
5mg
25mg
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TGX-115
Code: Asc-2078
Potent, selective, cell-permeable PI3-K inhibitor
>95%  
1mg
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TGX-221
Code: Asc-924
Potent, selective PI3K inhibitor
>98%  
100µg
500µg
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Thiazovivin
Code: Asc-2081
ROCK inhibitor. Fibroblast reprogramming efficiency enhancer.
>98%  
1mg
5mg
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TMCB
Code: Asc-289
Selective CK2 inhibitor
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10mg
50mg
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Triciribine
Code: Asc-936
Selective, potent inhibitor of Akt activation
>98%  
1mg
5mg
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7,3',4'-Trihydroxyisoflavone (7,3′,4′-THIF)
Code: Asc-1458
Isoflavone. Inhibits various kinase.
>98%  
25mg
100mg
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TWS119
Code: Asc-2075
Potent cell-permeable GSK-3β inhibitor
>95%  
2mg
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Tyrophostin AG1295
Code: Asc-2375
Selective PGDF receptor inhibitor
>98%  
1mg
5mg
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Tyrphostin 25 (RG-50875)
Code: Asc-1557
Competitive EGF receptor tyrosine kinase inhibitor
>99%  
5mg
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Tyrphostin 46 (AG-99)
Code: Asc-1571
EGF receptor tyrosine kinase inhibitor
>99%  
10mg
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Tyrphostin 47
Code: Asc-1558
EGFR tyrosine kinase inhibitor
>99%  
5mg
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Tyrphostin 51
Code: Asc-1559
EGFR tyrosine kinase inhibitor
>99%  
5mg
25mg
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Tyrphostin 9
Code: Asc-1561
Selective PDGFR tyrosine kinase inhibitor
>99%  
50mg
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Tyrphostin 8
Code: Asc-1731
Tyrosine kinase inhibitor
>98%  
10mg
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Tyrphostin AG 957
Code: Asc-1172
Potent, selective p210 tyrosine kinase inhibitor
>99%  
1mg
5mg
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U0126
Code: Asc-241
Selective MKK inhibitor
>98%  
5mg
25mg
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VX-702
Code: Asc-2057
Potent, selective p38 MAP kinase inhibitor
>99%  
1mg
5mg
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Wogonin
Code: Asc-2471
Cell permeable COX-2 inhibitor
>98%  
5mg
10mg
25mg
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Wortmannin
Code: Asc-148
PI3-kinase inhibitor
>98%  
1mg
5mg
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WP1066
Code: Asc-1440
JAK/STAT3 inhibitor; AG 490 analog
>97%  
5mg
25mg
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XRP44X
Code: Asc-1088
Cell-permeable Ras-Net (Elk-3) pathway inhibitor
>99%  
10mg
50mg
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Y-27632 dihydrochloride
Code: Asc-129
Selective Rho kinase inhibitor
>99%  
1mg
10mg
50mg
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YM201636
Code: Asc-1370
Potent, selective PIKfyve inhibitor
>95%  
1mg
5mg
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ZIP
Code: Asc-993
Novel, cell-permeable protein kinase Mζ (PKMζ) inhibitor
>97%  
1mg
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ZM 336372
Code: Asc-428
Potent, selective c-Raf inhibitor
>98%  
1mg
10mg
50mg
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